BET-IN-1 - CAS 1422554-34-4
Catalog number:
1422554-34-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H30N4O4
Molecular Weight:
450.53
COA:
Inquire
Targets:
BET Bromodomain
Description:
BET-IN-1, an oxazole derivative, can be used as a bromodomain inhibitor
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Appearance:
White to off-white Solid
Synonyms:
4-[8-methoxy-1-[(2R)-1-methoxypropan-2-yl]-2-(oxan-4-yl)imidazo[4,5-c]quinolin-7-yl]-3,5-dimethyl-1,2-oxazole BET-IN-1 SCHEMBL14698278 CS-5464 HY-19760
Solubility:
Soluble to ≥ 32 mg/mL in DMSO
Storage:
Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -34℃ for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years
Quantity:
Grams-Kilos
Boiling Point:
613.9±55.0 °C | Condition: Press: 760 Torr
InChIKey:
HYPXHDJBILNWLI-CQSZACIVSA-N
InChI:
1S/C25H30N4O4/c1-14(13-30-4)29-24-18-11-22(31-5)19(23-15(2)28-33-16(23)3)10-20(18)26-12-21(24)27-25(29)17-6-8-32-9-7-17/h10-12,14,17H,6-9,13H2,1-5H3/t14-/m1/s1
Canonical SMILES:
CC1=C(C(=NO1)C)C2=C(C=C3C(=C2)N=CC4=C3N(C(=N4)C5CCOCC5)C(C)COC)OC
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