BET bromodomain inhibitor - CAS 1505453-59-7
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C20H15Cl2N3O2
Molecular Weight:
400.259
COA:
Inquire
Targets:
BET Bromodomain
Description:
An BET bromodomain inhibitor can be used for the treatment of hematologic malignancies. It binds BET proteins to suppress the interaction between these proteins, propeins and acetylated chromatin, as well as transcription factors. The BET bromodomain inhibitor modulates the expression of oncogenes.
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Brife Description:
An BET bromodomain inhibitor, hematologic malignancies
Purity:
≥98%
Appearance:
Solid Powder
Synonyms:
2-[8-Chloro-6-(4-chloro-phenyl)-1-methyl-4H-3-oxa-2,5-diaza-benzo[e]azulen-4-yl]-acetamide
Solubility:
Soluble in DMSO.
Storage:
Store in a cool and dry place and at 0-4 ℃ for short term (days to weeks) or -66 ℃ for long term (months to years).
MSDS:
Inquire
Application:
the treatment of hematologic malignancies
Shelf Life:
2 years
InChIKey:
RKYPLOAYXFDLOF-UHFFFAOYSA-N
InChI:
InChI=1S/C20H15Cl2N3O2/c1-10-18-14-7-6-13(22)8-15(14)19(11-2-4-12(21)5-3-11)24-16(9-17(23)26)20(18)27-25-10/h2-8,16H,9H2,1H3,(H2,23,26)
Canonical SMILES:
CC1=NOC2=C1C3=C(C=C(C=C3)Cl)C(=NC2CC(=O)N)C4=CC=C(C=C4)Cl
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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