|Description||Bepotastine is a histamine H1 receptor antagonist. Bepotastine has been approved in Japan for the treatment of allergic rhinitis and uriticaria/puritus.|
|B0084-061917||500 mg||$248||In stock|
|Brife Description||Histamine H1 receptor antagonist|
|Related CAS||125602-71-3 (free base)|
|Synonyms||Bepotastine besylate; Bepreve; Betotastine besilate; Talion; 4-[(S)-(4-chlorophenyl)-2-pyridinylmethoxy]-1-piperidinebutanoic acid, monobenzenesulfonate|
PF-03654746 Tosylate is a histamine H3 receptor antagonist undergoing a clinical trial for attention-deficit hyperactivity disorder (ADHD) therapy.
JNJ 10181457 dihydrochloride
The hydrochloride salt form of JNJ 10181457, which has been found to be a histamine H3 receptor inhibitor and could be a brain penetrant.
Ebastine is a nonsedating type histamine H1-receptor antagonist.
Halopyramine is known as a competitive reversible H1-receptor antagonist. It exerts its pharmacological action by competing with histamine for the H1 subtype hi...
Famotine hydrochloride is a histamine H2 receptor antagonist. lt has no effect on the cytochrome P450 enzyme system, and does not appear to interact with other ...
Ketotifen is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators, used as self-medication for the temporary relief of ...
KDM5A-IN-1, a pyrrolidine amide compound, is an inhibitor histone demethylases.
A 943931 is a potent and selective histamine H4 receptor antagonist.
GS-283, an isoquinolin derivative, has been found to be histamine receptor and muscarinic receptor blocker.
CP66,948 is a histamine H2-receptor antagonist. It has gastric antisecretory activity and mucosal protective properties.
GT 2016 is a high affinity and brain-penetrant histamine H3 receptor antagonist (Ki = 43.8 nM). It displays selectivity against H1 and H2 receptors (IC50 >10 μM...
Lafutidine, a newly developed histamine H(2)-receptor antagonist, inhibits gastric acid secretion.
Levocabastine is a selective second-generation Histamine H1 receptor antagonist. It is used for Allergic conjunctivitis and Seasonal allergic rhinitis。Levocabas...
Thioperamide is a potent histamine H3 and H4 antagonist/inverse agonist (Ki = 25 and 27 nM for human recombinant H3 and H4 receptors, respectively). Thioperamid...
Diphenylpyraline, a piperidine derivative, has been found to be a H1 receptor antagonist that could be probably effective against some allergy acts.
LY-150310 is a histamine H1-receptor antagonist. It could alter prostanoid concentrations in vitro and in vivo.
A 987306 is a potent histamine H4 receptor antagonist (pKi = 8.24 and 8.47 in human and rat H4 receptors, respectively) with 162-, 620-, and > 1600-fold selecti...
Chlorpheniramine inhibits the proliferation of MCF-7, MDA-MB 231, and Ehrlich cells in a dose-response manner, and significantly reduces the ornithine decarboxy...
SUVN-G3031 is a Histamine H3 receptor antagonist originated by Suven Life Sciences. Blockade of Histamine H3 receptor can augment the pre-synaptic release of bo...
The hydrochloride salt form of Diphenylpyraline, one of the first-generation antihistamine agent, has been found to exhibit anticholinergic activity and could b...