BBI-503 - CAS 1129403-56-0
Catalog number: 1129403-56-0
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C31H33N5O2S
Molecular Weight:
539.69
COA:
Inquire
Targets:
Others
Description:
BBI-503 is a potent and selective CSCPK inhibitor with potential anticancer activity. It is an orally administered investigational agent designed to inhibit cancer stem cell pathways, including Nanog, by targeting stemness kinases.
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Purity:
>98%
Appearance:
Solid powder
Synonyms:
Amcasertib;BBI503;N-[2-(diethylamino)ethyl]-2,4-dimethyl-5-[(Z)-[2-oxo-5-(2-phenyl-1,3-thiazol-4-yl)-1H-indol-3-ylidene]methyl]-1H-pyrrole-3-carboxamide;(E)-N-(2-(diethylamino)ethyl)-2,4-dimethyl-5-((2-oxo-5-(2-phenylthiazol-4-yl)indolin-3-ylidene)methyl)-1H-pyrrole-3-carboxamide
Solubility:
DMSO ≥ 30 mg/Ml
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
BBI-503 has potential anticancer activity. It is designed to inhibit cancer stem cell pathways.
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Grams to Kilograms
Density:
1.246±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
QDWKGEFGLQMDAM-ULJHMMPZSA-N
InChI:
InChI=1S/C31H33N5O2S/c1-5-36(6-2)15-14-32-30(38)28-19(3)26(33-20(28)4)17-24-23-16-22(12-13-25(23)34-29(24)37)27-18-39-31(35-27)21-10-8-7-9-11-21/h7-13,16-18,33H,5-6,14-15H2,1-4H3,(H,32,38)(H,34,37)/b24-17-
Canonical SMILES:
CCN(CC)CCNC(=O)C1=C(NC(=C1C)C=C2C3=C(C=CC(=C3)C4=CSC(=N4)C5=CC=CC=C5)NC2=O)C
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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