Bazedoxifene acetate - CAS 198481-33-3
Catalog number:
198481-33-3
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C32H38N2O5
Molecular Weight:
530.66
COA:
Inquire
Targets:
Estrogen Receptor/ERR
Description:
Bazedoxifene acetate, also called as TSE424 or WAY-140424, with antiosteoporotic it is a selective nonsteroidal estrogen receptor modulator (SERM) (ERα: IC50= 26 nM; ERβ= 99 nM).
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Purity:
95%
Appearance:
Off-White to Pale Beige Solid.
Synonyms:
acetic acid;1-[[4-[2-(azepan-1-yl)ethoxy]phenyl]methyl]-2-(4-hydroxyphenyl)-3-methylindol-5-ol bazedoxifene bazedoxifene acetate TSE 424 TSE-424 TSE424 WAY-140424
Solubility:
Soluble to 5.2 mg/mL in DMSO
Storage:
Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -29℃ for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years
Quantity:
Data not available, please inquire.
Boiling Point:
694.4ºC at 760 mmHg
InChIKey:
OMZAMQFQZMUNTP-UHFFFAOYSA-N
InChI:
1S/C30H34N2O3.C2H4O2/c1-22-28-20-26(34)12-15-29(28)32(30(22)24-8-10-25(33)11-9-24)21-23-6-13-27(14-7-23)35-19-18-31-16-4-2-3-5-17-31;1-2(3)4/h6-15,20,33-34H,2-5,16-19,21H2,1H3;1H3,(H,3,4)
Canonical SMILES:
CC1=C(N(C2=C1C=C(C=C2)O)CC3=CC=C(C=C3)OCCN4CCCCCC4)C5=CC=C(C=C5)O.CC(=O)O
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Chemical Structure

CAS 198481-33-3 Bazedoxifene acetate

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