Bavisant - CAS 929622-08-2
Catalog number: 929622-08-2
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H27N3O2
Molecular Weight:
329.44
COA:
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Targets:
Histamine Receptor
Description:
Bavisant is a highly selective, orally active antagonist of the human H3 receptor. It is a novel mechanism of action, involving wakefulness and cognition. It has potential to be used as a treatment for ADHD. It was developed by Johnson & Johnson and has completed a phase II ADHD trial, but there has been no progress.
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Purity:
>98%
Appearance:
Solid powder
Synonyms:
JNJ 31001074;JNJ-31001074;(4-Cyclopropylpiperazin-1-yl)-[4-(morpholin-4-ylmethyl)phenyl]methanone
Solubility:
10 mM in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Bavisant has potential to be used as a treatment for ADHD.
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
Boiling Point:
485.2±45.0 °C | Condition: Press: 760 Torr
Density:
1.220±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
BGBVSGSIXIIREO-UHFFFAOYSA-N
InChI:
InChI=1S/C19H27N3O2/c23-19(22-9-7-21(8-10-22)18-5-6-18)17-3-1-16(2-4-17)15-20-11-13-24-14-12-20/h1-4,18H,5-15H2
Canonical SMILES:
C1CC1N2CCN(CC2)C(=O)C3=CC=C(C=C3)CN4CCOCC4
Current Developer:
Bavisant was developed by Johnson & Johnson and has completed a phase II ADHD trial, but there has been no progress.
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CAS 929622-08-2 Bavisant

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