Barnetil - CAS 53583-79-2
Catalog number: 53583-79-2
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C17H26N2O4S
Molecular Weight:
354.46
COA:
Inquire
Targets:
Dopamine Receptor
Description:
Barnetil acts as a selective D2 and D3 receptor antagonist, which has high affinity for these receptors of dissociation constants of 2.2 nM and 2.4 nM respectively. It is an atypical antipsychotic used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder. It has also been shown to have clinically relevant affinity for the GHB receptor. It was launched by Sanofi-Aventis in 1976.
Publictions citing BOC Sciences Products
  • >> More
Purity:
98%
Appearance:
Solid powder
Synonyms:
Sultopride;Benzamide, N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-(ethylsulfonyl)-2-methoxy- (9CI);N-[(1-Ethyl-2-pyrrolidinyl)methyl]-5-(ethylsulfonyl)-2-methoxybenzamide;N-[(1-Ethylpyrrolidin-2-yl)methyl]-5-(ethylsulfonyl)-2-(methyloxy)benzamide
Solubility:
Soluble in DMSO, not in water
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Barnetil is used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder.
Quality Standard:
In-house standard
Quantity:
Kilograms to Tons
Boiling Point:
530.0±50.0 °C | Condition: Press: 760 Torr
Melting Point:
181-182 °C
Density:
1.160±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
UNRHXEPDKXPRTM-UHFFFAOYSA-N
InChI:
InChI=1S/C17H26N2O4S/c1-4-19-10-6-7-13(19)12-18-17(20)15-11-14(24(21,22)5-2)8-9-16(15)23-3/h8-9,11,13H,4-7,10,12H2,1-3H3,(H,18,20)
Canonical SMILES:
CCN1CCCC1CNC(=O)C2=C(C=CC(=C2)S(=O)(=O)CC)OC
Current Developer:
Barnetil was launched by Sanofi-Aventis in 1976.
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related Dopamine Receptor Products


CAS 91374-20-8 Ropinirole HCl

Ropinirole HCl
(CAS: 91374-20-8)

Ropinirole a selective D-2 agonist with Ki of 29 nM.

CAS 1148156-63-1 ST-836

ST-836
(CAS: 1148156-63-1)

ST-836, a dopamine receptor ligand, might have similar effect with dopamine and probably useful as an antiparkinsonian agent.

CAS 269718-84-5 Pardoprunox

Pardoprunox
(CAS: 269718-84-5)

Pardoprunox, also called as SLV308 or DU-126891, is a D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist (IA = 50% and 67%, respectively) and 5-HT1A rec...

CAS 34161-24-5 Fipexide

Fipexide
(CAS: 34161-24-5)

Fipexide hydrochloride is a nootropic agent that displays a positive effect on cognitive function

CAS 108050-82-4 Roxindole hydrochloride

Roxindole hydrochloride
(CAS: 108050-82-4)

Roxindole hydrochloride is a selective and potent presynaptic D-2 dopamine autoreceptor agonist, with affinity for D3, D4 and 5-HT1 receptors (pKi values are 8....

CAS 97612-24-3 Eticlopride hydrochloride

Eticlopride hydrochloride
(CAS: 97612-24-3)

Eticlopride hydrochloride is a selective dopamine D2/D3 receptor antagonist (Ki = 0.50 and 0.16 nM, respectively).

CAS 189744-94-3 Ro 10-5824 dihydrochloride

Ro 10-5824 dihydrochloride
(CAS: 189744-94-3)

Ro 10-5824, a D4R partial agonist, might have beneficial effects on attention and impulsivity by modulating baseline gamma activity in the frontal cortex.

CAS 1227675-51-5 SCH 39166 hydrobromide

SCH 39166 hydrobromide
(CAS: 1227675-51-5)

SCH 39166 hydrobromide is a high affinity dopamine D1/D5 receptor antagonist (Ki = 1.2, 2, 980, 5520, 80 and 731 nM for binding to D1, D5, D2, D4, 5-HT and α2a ...

CAS 114200-31-6 PAOPA

PAOPA
(CAS: 114200-31-6)

PAOPA is an allosteric modulator of dopamine D2 receptors. It can prevent and reverse behavioral and biochemical abnormalities in an amphetamine-sensitized anim...

Haloperidol hydrochloride
(CAS: 1511-16-6)

Haloperidol hydrochloride is a dopamine antagonist that specifically targets D2-like receptors, with effect to treat schizophrenia, acute psychosis, and deliriu...

CAS 53772-83-1 Zuclopenthixol

Zuclopenthixol
(CAS: 53772-83-1)

Zuclopenthixol is an antagonist at D1 and D2 dopamine receptors. It also has high affinity for alpha1-adrenergic and 5-HT2 receptors, but it has weaker histamin...

CAS 2022-29-9 Spiperone hydrochloride

Spiperone hydrochloride
(CAS: 2022-29-9)

Spiperone hydrochloride is a 5-HT2A and selective dopamine D2 receptor antagonist (Ki = 0.06, 0.6, 0.08, ~ 350, ~ 3500 nM for D2, D3, D4, D1 and D5 receptors, r...

CAS 200954-39-8 Dilept

Dilept
(CAS: 200954-39-8)

Dilept is an antagonist of neurotensin (NT) and dopamine (DA) receptor used to mitigate positive and negative symptoms of schizophrenia.

CAS 93601-85-5 (R)-5-Methoxy-N-propyl-2-aminotetraline hydrochloride

(R)-5-Methoxy-N-propyl-2-aminotetraline
(CAS: 93601-85-5)

(R)-5-Methoxy-N-propyl-2-Aminotetraline hydrochloride is a dopamine receptor agonist and an intermediate in the production of antipsychotic agents and antiparki...

CAS 32672-69-8 Mesoridazine besylate

Mesoridazine besylate
(CAS: 32672-69-8)

Mesoridazine besylate, a phenothiazine dopamine receptor anatagonist, has been described to demonstrate inhibition for D2DR and D4DR. High affinity for the clon...

CAS 23257-56-9 Levophacetoperane hydrochloride

Levophacetoperane hydrochloride
(CAS: 23257-56-9)

Levophacetoperane hydrochloride, a sympathomimetic central nervous system stimulant used to treat depression, inhibits in vitro in a competitive manner, norepin...

CAS 300561-58-4 SKF 77434 hydrobromide

SKF 77434 hydrobromide
(CAS: 300561-58-4)

SKF 77434 hydrobromide is a selective dopamine D1-like receptor partial agonist (IC50 = 19.7 and 2425 nM for binding to D1-like and D2-like receptors, respectiv...

CAS 123240-93-7 R(-)-N-Ethylnorapomorphine hydrochloride

R(-)-N-Ethylnorapomorphine hydrochloride
(CAS: 123240-93-7)

R(-)-N-Ethylnorapomorphine hydrochloride is a dopamine D2 receptor agonist.

CAS 36085-44-6 B-HT 958 dihydrochloride

B-HT 958 dihydrochloride
(CAS: 36085-44-6)

B-HT 958 dihydrochloride is a dopamine D2 receptor agonist and an α2-adrenoceptor partial agonist.

CAS 67383-44-2 RU 24213

RU 24213
(CAS: 67383-44-2)

RU 24213 is a dopamine D2 receptor agonist as well as a kappa opioid receptor antagonist.

Chemical Structure

CAS 53583-79-2 Barnetil

Quick Inquiry

Verification code

Featured Items