Barnetil - CAS 53583-79-2
Catalog number: 53583-79-2
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C17H26N2O4S
Molecular Weight:
354.46
COA:
Inquire
Targets:
Dopamine Receptor
Description:
Barnetil acts as a selective D2 and D3 receptor antagonist, which has high affinity for these receptors of dissociation constants of 2.2 nM and 2.4 nM respectively. It is an atypical antipsychotic used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder. It has also been shown to have clinically relevant affinity for the GHB receptor. It was launched by Sanofi-Aventis in 1976.
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Purity:
98%
Appearance:
Solid powder
Synonyms:
Sultopride;Benzamide, N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-(ethylsulfonyl)-2-methoxy- (9CI);N-[(1-Ethyl-2-pyrrolidinyl)methyl]-5-(ethylsulfonyl)-2-methoxybenzamide;N-[(1-Ethylpyrrolidin-2-yl)methyl]-5-(ethylsulfonyl)-2-(methyloxy)benzamide
Solubility:
Soluble in DMSO, not in water
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Barnetil is used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder.
Quality Standard:
In-house standard
Quantity:
Kilograms to Tons
Boiling Point:
530.0±50.0 °C | Condition: Press: 760 Torr
Melting Point:
181-182 °C
Density:
1.160±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
UNRHXEPDKXPRTM-UHFFFAOYSA-N
InChI:
InChI=1S/C17H26N2O4S/c1-4-19-10-6-7-13(19)12-18-17(20)15-11-14(24(21,22)5-2)8-9-16(15)23-3/h8-9,11,13H,4-7,10,12H2,1-3H3,(H,18,20)
Canonical SMILES:
CCN1CCCC1CNC(=O)C2=C(C=CC(=C2)S(=O)(=O)CC)OC
Current Developer:
Barnetil was launched by Sanofi-Aventis in 1976.
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CAS 53583-79-2 Barnetil

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