|Description||Bambuterol is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma.|
Lusaperidone, also known as R107474, is an α2 adrenergic receptor antagonist. R107474 showed high affinity for ha2A-, ha2B-, and ha2C-adrenoceptors, stably expr...
Fenspiride is an α adrenergic and H1 histamine receptor antagonist. It is an oxazolidinone spiro compound. It is used as a drug in the treatment of certain resp...
Atenolol, with antianginal and antiarrhythmic properties, it is a cardioselective beta-adrenergic blocker and used in hypertension control.
Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM, used as a "reliever" inhaler in the management of asthma symptoms and as a...
Penbutolol is a sympathomimetic drug used to treat mild to moderate high blood pressure by binding to both beta-1 adrenergic receptors and beta-2 adrenergic rec...
Tetrahydrozoline HCl is an imidazoline derivative with alpha receptor agonist activity.
Isoprenaline is a non-selective beta-adrenergic receptor agonist, used for the treatment of bradycardia and heart block. It would increase cAMP levels and activ...
Tolazoline is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn..
Xylometazoline is an α-adrenoceptor agonist commonly used as nasal decongestant, exhibits highest potency at α2B-adrenoceptor subtype with EC50 of 99 μM.
Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation.
CP-331684 is a β3-adrenergic receptor agonist used as antidiabetic drug.
Aptazapine is a tetracyclic antidepressant. It was assayed in clinical trials for the treatment of depression in the 1980s but was never marketed. Aptazapine is...
The hydrochloride of Nifenalol. Nifenalol is a beta-adrenoceptor antagonist used for the treatment of cardiovascular and cerebrovascular diseases such as hypert...
Naftopidil is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM.
Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
Levosalbutamol tartrate, the R-enantiomer of salbutamol, is a short-acting β2 adrenergic receptor agonist used in the treatment of asthma and chronic obstructiv...
BMS-196085, a sulfanilamide derivative, has been found to be a β-adrenergic receptor agonist that was once studied in obesity as well as yype 2 diabetes mellitu...
(R,R)-Formoterol is a long acting beta-adrenoceptor agonist acts as a novel highly β2-selective adrenergic agonist and holds promise as a β2-agonist that could ...
Rauwolscine hydrochloride is the hydrochloride salt of Rauwolscine which is a potent, reversible and specific α2 adrenergic receptor antagonist with a Ki values...
Silodosin shows high selectivity for the alpha(1A)-AR subtype.