|Description||BAMB-4 is a new membrane-permeable inhibitor against inositol-1,4,5-trisphosphate-3-kinase A((ITPKA). It exhibits the lowest inhibition frequency among the InsP3-Kinase inhibitors. It is a promising therapeutic approach in lung cancer therapy.|
Exhibits high affinity for TSPO in rat whole brain (Ki = 0.297 nM), and high potency against human and rat glial TSPO (IC50 values are 2.73 and 3.04 nM respecti...
Chlormezanone, a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.
GI 254023X is a selective ADAM10 metalloprotease inhibitor with over 100-fold higher potency at ADAM10 than ADAM17. GI 254023X inhibits the proliferation of H92...
Ritobegron ethyl hydrochloride
Ritobegron is a potential Bladder selectivity of the novel β₃-agonist.
JNJ 63533054 is a potent and selective GPR139 agonist (EC50 = 16 nM) that is brain and cell penetrant. JNJ 63533054 is selective for GPR139 over a panel of GPCR...
Izonsteride, a benzothiazolyl derivative, has been found to be a cholestenone 5-alpha reductase inhibitor that was once studied in prostate cancer and probably ...
This active molecular is a selective Porcupine protein inhibitor and IC50 value is 0.8nM. GNF-6231 shows efficient pathway inhibition and induced robust antitum...
Namiteca is a new water-soluble camptothecin analogue as a hydrophilic camptothecin with a promising preclinical profile.
Pyrintegrin, a 2,4-disubstituted pyrimidine, enhances survival of human embryonic stem cells (hESCs) following enzymatic dissociation. Pyrintegrin increases the...
A impurity of Desogestrel, which is a progestogen.
Miglustat is an inhibitor of the ceramide-specific glycosyltransferase, which catalyzes the first step of glycosphingolipid biosynthesis and is currently approv...
all cis-5,8,11,14,17-Eicosapentaenoic Ac
all cis-5,8,11,14,17-Eicosapentaenoic Acid Ethyl Ester is an omega-3 fatty acid agent. It is important polyunsaturated fatty acid of the marine food chain. It s...
CP-5068 is a synthetic bio-active chemical.
3-Methylsalicylic acid has marked fibrinolytic activity in human plasma by activating its fibrinolytic system. It is a salicylic acid derivative compound, which...
HL 010183 is a metformin derivative exhibiting potent antitumor effect. It inhibits proliferation and invasion of Hs578T triple-negative (TN) breast cancer cell...
GSK 264220A is an endothelial lipase and lipoprotein lipase inhibitor (IC50 = 0.13 and 0.10 μM, respectively). Inhibition of endothelial lipase may lead to an i...
NITD008 is a flavivirus inhibitor. It was developed as a potential treatment for flavivirus infections, and shows broad spectrum antiviral activity.
Pozanicline, a pyridine derivative, has been found to be a nicotinic receptor modulator that was once studied in Alzheimer's disease as a neuroprotective agent.
Fmoc-Val-Cit-PAB-PNP is a peptide prodrug linker. It is a linker for antibody-drug-conjugation (ADC).
Bisacodyl (INN) is a stimulant laxative drug that works directly on the colon to produce a bowel movement.Bisacodyl works by stimulating enteric nerves to cause...