AZD9496 - CAS 1639042-08-2
Catalog number: B0084-470890
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H25F3N2O2
Molecular Weight:
442.48
COA:
Inquire
Targets:
Estrogen Receptor/ERR
Description:
AZD9496 is a potent and orally bioavailable selective estrogen receptor downregulator and antagonist. AZD9496 can induce ERα degradation in breast cancer cell lines at picomolar concentrations.
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-470890 25 mg $198 In stock
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Purity:
98%
Related CAS:
1639042-28-6 (maleate)
Appearance:
Solid powder
Synonyms:
(E)-3-(3,5-difluoro-4-((1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)phenyl)acrylic acid; AZD9496; AZD-9496; AZD 9496
Solubility:
Soluble in DMSO, not in water
Storage:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years if stored properly
InChIKey:
DFBDRVGWBHBJNR-BBNFHIFMSA-N
InChI:
1S/C25H25F3N2O2/c1-14-10-17-16-6-4-5-7-20(16)29-23(17)24(30(14)13-25(2,3)28)22-18(26)11-15(12-19(22)27)8-9-21(31)32/h4-9,11-12,14,24,29H,10,13H2,1-3H3,(H,31,32)/b9-8+/t14-,24-/m1/s1
Canonical SMILES:
O=C(O)/C=C/C1=CC(F)=C([C@H]2N(CC(C)(F)C)[C@H](C)CC3=C2NC4=C3C=CC=C4)C(F)=C1
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CAS 1639042-08-2 AZD9496

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