AZD1979 - CAS 1254035-84-1
Catalog number: 1254035-84-1
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H26N4O5
Molecular Weight:
462.51
COA:
Inquire
Targets:
MCH1
Description:
This active molecular is a MCHr1 (melanin concentrating hormone receptor 1) antagonist originated by AstraZeneca. AZD1979 has excellent DMPK properties and gave good effects on weight loss in animal model. In Jul 2014, AstraZeneca terminated a phase I trial in Obesity in healthy volunteers in USA after stopping criteria were reached .
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Purity:
98%
Appearance:
Powder
Synonyms:
(3-(4-((2-oxa-6-azaspiro[3.3]heptan-6-yl)methyl)phenoxy)azetidin-1-yl)(5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl)methanone
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Obesity
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
Canonical SMILES:
O=C(N1CC(OC2=CC=C(CN(C3)CC43COC4)C=C2)C1)C5=NN=C(C6=CC=C(OC)C=C6)O5
Current Developer:
Originator:AstraZeneca
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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