|Description||The (-)-enantiomer of Azasetron hydrochloride, which is a selective 5-HT3 antagonist.|
|Brife Description||5-HT3 antagonist|
|Related CAS||123040-16-4 (racemic)|
Fananserin is a 5-HT2A receptor and a dopamine D4 receptor antagonist (Ki = 0.26, 2.93, 25, 38, 70 and 726 nM for 5-HT2A, D4, H1, α1, 5-HT1A and D2 receptors, r...
Agomelatine is a melatoninergic agonist and selective antagonist of 5-HT2C receptors, and has been shown to be active in several animal models of depression. Ag...
SB 258585 hydrochloride
SB 258585 hydrochloride is a potent and selective 5-HT6 receptor antagonist (pKi = 8.6) with > 160-fold selectivity over other 5-HT receptor subtypes, dopamine ...
MS 245 oxalate
MS 245 oxalate is a 5-HT6 antagonist with high affinity (Ki = 2.1 nM). It potentiates the hypolocomotor actions of (-)-nicotine in mice.
Methysergide is an ergot derivative that is a congener of lysergic acid diethylamide for the treatment of vascular headache
PNU 22394 hydrochloride
PNU 22394 is virtually a full agonist at 5-HT2C receptors (87% of 5-HT), but a partial agonist at 5-HT2A (65% of 5-HT), and 5-HT2B (<15% of 5-HT) receptors. It ...
Granisetron HCl is a serotonin 5-HT3 receptor antagonist.
SB 242084 is a brain-penetrant antagonist of 5-HT2C receptor which exhibits 158-fold selectivity for 5-HT2C (pKi= 9.0) over 5-HT2A receptor (pKi= 6.1-6.8) and 1...