|Description||The (+)-enantiomer of Azasetron hydrochloride, which is a selective 5-HT3 antagonist.|
|Brife Description||5-HT3 antagonist|
|Related CAS||123040-16-4 (racemic)|
SB 242084 is a brain-penetrant antagonist of 5-HT2C receptor which exhibits 158-fold selectivity for 5-HT2C (pKi= 9.0) over 5-HT2A receptor (pKi= 6.1-6.8) and 1...
RS 127445 hydrochloride
RS-127445 is a selective, high affinity, orally bioavailable serotonin 5-HT2B receptor antagonist (pKi = 9.5), which displays 1000-fold selectivity for 5-HT2B w...
SB 258719 hydrochloride
SB 258719 hydrochloride is a selective 5-HT7 receptor antagonist, displaying > 100-fold selectivity over a range of other receptors. SB 258719 shows inverse act...
Quetiapine sulfoxide dihydrochloride
Quetiapine sulfoxide dihydrochloride, a metabolite of Quetiapine, has antipsychotic effect.
LP 20 hydrochloride
LP 20 hydrochloride is a ligand of the 5-HT7 receptor. It shows agonist and antagonist activity.
LY 393558 is a 5-HT reuptake inhibitor with pIC50 value of 8.48. It is also a dual 5-HT1B/1D receptor antagonist with pKB values of 9.05 and 8.98 respectively.
Anpirtoline hydrochloride is the hydrochloride salt of anpirtoline, which is a highly potent 5-HT1B receptor agonist with Ki values of 28 nM. It decreases centr...
Way 100135 is a selective 5-HT1A receptor antagonist originated by Wyeth with IC50 value of 15 nM. IC 50 values for 5-HT1B, 1C, 2,α1, α2 and D2 receptors are ov...