AZ0108 - CAS 1825345-52-5
Catalog number: 1825345-52-5
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C24H20F4N6O2
Molecular Weight:
500.45
COA:
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Targets:
PARP
Description:
AZ0108 is an orally bioavailable, PARP1,2,6 inhibitor that causes a multi-polar spindle phenotype at double digit nM concentrations. AZ0108 has been utilized as in vitro tools and in vivo probes to investigate the biological consequences of inhibiting centrosome clustering through PARP enzymes.
Purity:
>98%
Appearance:
Solid powder
Synonyms:
(S)-4-((3-(3-(1,1-difluoroethyl)-6-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl)phenyl)difluoromethyl)phthalazin-1(2H)-one; AZ0108; AZ-0108; AZ 0108.
MSDS:
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Canonical SMILES:
O=C1NN=C(C2=CC=CC=C21)C(F)(F)C3=CC=CC(C(N4[C@@H](C)CN5C(C4)=NN=C5C(F)(F)C)=O)=C3
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