AZ0108 - CAS 1825345-52-5
Catalog number:
1825345-52-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C24H20F4N6O2
Molecular Weight:
500.45
COA:
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Targets:
PARP
Description:
AZ0108 is an orally bioavailable, PARP1,2,6 inhibitor that causes a multi-polar spindle phenotype at double digit nM concentrations. AZ0108 has been utilized as in vitro tools and in vivo probes to investigate the biological consequences of inhibiting centrosome clustering through PARP enzymes.
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Purity:
>98%
Appearance:
Solid powder
Synonyms:
(S)-4-((3-(3-(1,1-difluoroethyl)-6-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl)phenyl)difluoromethyl)phthalazin-1(2H)-one; AZ-0108; AZ 0108
MSDS:
Inquire
Canonical SMILES:
O=C1NN=C(C2=CC=CC=C21)C(F)(F)C3=CC=CC(C(N4[C@@H](C)CN5C(C4)=NN=C5C(F)(F)C)=O)=C3
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