|Description||AT 1001 is a partial agonist and antagonist of α3β4 nAChR ligand (Ki value 2.6 nM at α3β4 nAChR). In vivo AT-1001 potently blocks nicotine self-administration in dose manner.|
|Brife Description||α3β4 nAChR inhibitor|
|Synonyms||AT 1001; AT1001; AT-1001|
5-Iodo-A-85380 dihydrochloride is the dihydrochloride salt of 5-Iodo-A-85380, which is a highly potent and subtype-selective agonist for α4β2 and α6β2 nicotinic...
α-Conotoxin MII is a nicotinic acetylcholine receptor antagonist. It is highly potent, selective and competitive for α3β2 subunit. Its IC50 value is 0.5-3.5 nM ...
4-Acetyl-1,1-dimethylpiperazinium iodide is a structural analog of acetylcholine, which is a nicotinic (AChR) agonist with Ki value of 29.9 nM at α4β2.
AZD 0328 is a potent α7 NNR/5HT3 receptor agonist. AZD0328 led to a significant increase in cortical dopamine release in awake rodents and improved both conditi...
Decamethonium Bromide is a nicotinic AChR partial agonist and neuromuscular blocking agent.
The hydrochloride salt form of α-Lobeline, a nicotinic receptor agonist, could be used against asphyxia and respiratory failure.
Tebanicline hydrochloride is the hydrochloride salt of Tebanicline (ABT-594) which is a neuronal nicotinic acetyl-choline receptor agonist and has been describe...
SIB 1553A hydrochloride
SIB 1553A hydrochloride is a nicotinic acetylcholine receptor (nAChR) agonist with selectivity for β4 subunit-containing receptors. It stimulates acetylcholine ...