ASP-8497 - CAS 651055-26-4
Catalog number:
651055-26-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C18H27FN4O7S
Molecular Weight:
462.49
COA:
Inquire
Targets:
DPP4
Description:
ASP8497 is a long-acting and potent DPP-IV inhibitor. It improves glucose tolerance through glucose-dependent insulinotropic action via elevation of the GLP-1 level. It is used as a therapeutic agent for impaired glucose tolerance and type 2 diabetes.
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Purity:
98%
Appearance:
Solid powder
Synonyms:
2-Pyrrolidinecarbonitrile, 4-fluoro-1-(((4-methyl-1-(methylsulfonyl)-4-piperidinyl)amino)acetyl)-, (2S,4S)-(2E)-2-butenedioate (1:1);ASP8497;(E)-but-2-enedioic acid (2S,4S)-4-fluoro-1-[2-[(4-methyl-1-methylsulfonylpiperidin-4-yl)amino]acetyl]pyrrolidine-2
Solubility:
Soluble in DMSO, not in water
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
ASP8497 is used as a therapeutic agent for impaired glucose tolerance and type 2 diabetes.
Quality Standard:
In-house standard
Quantity:
Milligrams-Grams
InChIKey:
YZYBLEWOKAXTOL-QPPPMHOJSA-N
InChI:
InChI=1S/C14H23FN4O3S.C4H4O4/c1-14(3-5-18(6-4-14)23(2,21)22)17-9-13(20)19-10-11(15)7-12(19)8-16;5-3(6)1-2-4(7)8/h11-12,17H,3-7,9-10H2,1-2H3;1-2H,(H,5,6)(H,7,8)/b;2-1+/t11-,12-;/m0./s1
Canonical SMILES:
CC1(CCN(CC1)S(=O)(=O)C)NCC(=O)N2CC(CC2C#N)F.C(=CC(=O)O)C(=O)O
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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