Asimadoline - CAS 153205-46-0
Catalog number: B0084-071264
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C27H30N2O2
Molecular Weight:
414.549
COA:
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Targets:
Opioid Receptor
Description:
Asimadoline is a κ opioid receptor agonist with less brain-penetrant ability. Asimadoline is the potential treatment of irritable bowel syndrome.
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-071264 50 mg $399 In stock
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Brife Description:
κ opioid receptor (KOR) agonist
Synonyms:
N-[(1S)-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-phenylethyl]-N-methyl-2,2-diphenylacetamide
Solubility:
DMSO: ≥ 103.3 mg/mL (249.19 mM)
MSDS:
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Boiling Point:
605.8±55.0 °C at 760 mmHg
Density:
1.2±0.1 g/cm3
InChIKey:
JHLHNYVMZCADTC-LOSJGSFVSA-N
InChI:
InChI=1S/C27H30N2O2/c1-28(25(21-11-5-2-6-12-21)20-29-18-17-24(30)19-29)27(31)26(22-13-7-3-8-14-22)23-15-9-4-10-16-23/h2-16,24-26,30H,17-20H2,1H3/t24-,25+/m0/s1
Canonical SMILES:
CN(C(CN1CCC(C1)O)C2=CC=CC=C2)C(=O)C(C3=CC=CC=C3)C4=CC=CC=C4
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Chemical Structure

CAS 153205-46-0 Asimadoline

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