AS-252424 - CAS 900515-16-4
Catalog number: 900515-16-4
Category: Inhibitor
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Molecular Formula:
C14H8FNO4S
Molecular Weight:
305.28
COA:
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Targets:
PI3K
Description:
AS-252424 is a novel, potent PI3Kγ inhibitor (IC50 of 30 nM) with a 30-fold selectivity for PI3Kγ than PI3Kα, and low inhibitory activity towards PI3Kδ/β.
Purity:
>98%
Synonyms:
AS252424; AS 252424; AS-252424.
MSDS:
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InChIKey:
OYYVWNDMOQPMGE-SDQBBNPISA-N
InChI:
InChI=1S/C14H8FNO4S/c15-7-1-3-9(10(17)5-7)11-4-2-8(20-11)6-12-13(18)16-14(19)21-12/h1-6,17H,(H,16,18,19)/b12-6-
Canonical SMILES:
C1=CC(=C(C=C1F)O)C2=CC=C(O2)C=C3C(=O)NC(=O)S3
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