AS-1669058 - CAS 1395553-31-7
Catalog number:
1395553-31-7
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C18-H15-Br-F2-N4-O
Molecular Weight:
421.24
COA:
Inquire
Targets:
GPR119
Description:
AS-1669058 is a G-protein-coupled receptor 119 (GPR119) agonist originated by Astellas Pharma. No recent reports of development were identified for preclinical development in Type-2-diabetes-mellitus in Japan.
Publictions citing BOC Sciences Products
  • >> More
Purity:
98%
Appearance:
Powder
Synonyms:
3-(2-((2-(4-bromo-2,5-difluorophenyl)-6-methylpyrimidin-4-yl)amino)ethyl)pyridine 1-oxide;AS 1535907; AS 1669058; AS 1907417; GPR119 agonists - Astellas Pharma;1395553-32-8(OXLATE)
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Type 2 diabetes mellitus
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
CCHGKGFZEORIJY-UHFFFAOYSA-N
InChI:
1S/C18H15BrF2N4O/c1-11-7-17(22-5-4-12-3-2-6-25(26)10-12)24-18(23-11)13-8-16(21)14(19)9-15(13)20/h2-3,6-10H,4-5H2,1H3,(H,22,23,24)
Canonical SMILES:
Cc1cc(nc(n1)c2cc(c(cc2F)Br)F)NCCc3ccc[n+](c3)[O-]
Current Developer:
Originator Astellas Pharma
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related GPR119 Products


CAS 832714-46-2 APD668

APD668
(CAS: 832714-46-2)

APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119 respectively.

APD597 (JNJ-38431055)
(CAS: 897732-93-3)

APD597, also known as JNJ-38431055, is a potent and selective GPR119 agonist, which is potential useful for the treatment of type 2 diabetes. GPR119 agonists me...

CAS 1032823-75-8 GSK-1292263

GSK-1292263
(CAS: 1032823-75-8)

GSK1292263 is a novel GPR119 receptor agonist used for the treatment of type 2 diabetes.

AS-1669058 oxalate
(CAS: 1395553-32-8)

AS-1669058 is a G-protein-coupled receptor 119 (GPR119) agonist originated by Astellas Pharma. No recent reports of development were identified for preclinical ...

CAS 733750-99-7 AR 231453

AR 231453
(CAS: 733750-99-7)

AR231453 is a potent and selective small molecule agonist of GPR119 that enhances glucose-dependent insulin secretion and glucagon-like peptide 1 (GLP-1) releas...

BMS 903452
(CAS: 1339944-47-6)

G-protein-coupled receptor 119 agonists can stimulate glucose-dependent insulin release by direct action in the pancreas and promote secretion of the incretin G...

CAS 857652-30-3 PSN632408

PSN632408
(CAS: 857652-30-3)

PSN632408 is an optimized agonist of GPR119 receptors that shows similar potency to OEA at both recombinant mouse and human GPR119 receptors. It suppresses food...

AS-1669058
(CAS: 1395553-31-7)

AS-1669058 is a G-protein-coupled receptor 119 (GPR119) agonist originated by Astellas Pharma. No recent reports of development were identified for preclinical ...

CAS 1037792-44-1 MBX-2982

MBX-2982
(CAS: 1037792-44-1)

MBX-2982 is a potential first-in-class treatment for type 2 diabetes that targets G protein-coupled receptor 119 (GPR119), a receptor that interacts with bioact...

Quick Inquiry

Verification code

Featured Items