Argipressine - CAS 113-79-1
Catalog number:
113-79-1
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C46H65N15O12S2
Molecular Weight:
1084.23
COA:
Inquire
Targets:
Vasopressin Receptor
Description:
This molecular is a polypeptide which is a Antidiuretic hormone that has been found in most mammalian species and it acts as a neurotransmitter at synapses in the brain to increases[Ca2+]i in cultured rat hippocampal neurons. In the Past, Arg-vasopressin was applicated to treat diabetes insipidus or to improve vasomotor tone and blood pressure. In 2008, preclinical trials in Heart was failed in USA (Intranasal).
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Purity:
95%
Appearance:
White powder
Synonyms:
H-Cys(1)-Tyr-Phe-Gln-Asn-Cys(1)-Pro-Arg-Gly-NH2,(2S)-1-[(4R,7S,10S,13S,16S,19R)-19-amino-7-(2-amino-2-oxoethyl)-10-(3-amino-3-oxopropyl)-13-benzyl-16-[(4-hydroxyphenyl)methyl]-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carbonyl]-N-[(2S)-1-[(2-amino-2-oxoethyl)amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]pyrrolidine-2-carboxamide
Solubility:
0.50 mg/ml in H2O
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
treat diabetes insipidus or to improve vasomotor tone and blood pressure
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
KBZOIRJILGZLEJ-LGYYRGKSSA-N
InChI:
InChI=1S/C46H65N15O12S2/c47-27-22-74-75-23-33(45(73)61-17-5-9-34(61)44(72)56-28(8-4-16-53-46(51)52)39(67)54-21-37(50)65)60-43(71)32(20-36(49)64)59-40(68)29(14-15-35(48)63)55-41(69)31(18-24-6-2-1-3-7-24)58-42(70)30(57-38(27)66)19-25-10-12-26(62)13-11-25/h1
Canonical SMILES:
C1CC(N(C1)C(=O)C2CSSCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N2)CC(=O)N)CCC(=O)N)CC3=CC=CC=C3)CC4=CC=C(C=C4)O)N)C(=O)NC(CCCN=C(N)N)C(=O)NCC(=O)N
Current Developer:
Originator: DelSite Biotechnologies
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CAS 113-79-1 Argipressine

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