|Description||ARC239 dihydrochloride is a potent and selective α2 B adrenoceptor antagonist. It is used as an α-adrenoceptor blocking drug. It competitively antagonizes pressor responses to adrenaline and inhibits pressor responses to noradrenaline, tyramine, phenylephrine and dimethylphenylpiperazinium.|
|Synonyms||2-(2-(4-(2-Methoxyphenyl)piperazin-1-yl)ethyl)-4,4-dimethyl-1,3-(2H,4H)-isoquinolindione dihydrochloride;AR-C239 Dihydrochloride|
|Solubility||Soluble in DMSO, not in water|
|Application||ARC239 dihydrochloride is used as an α-adrenoceptor blocking drug.|
|Quality Standard||In-house standard|
|Boiling Point||595.8±50.0 °C | Condition: Press: 760 Torr|
|Density||1.167±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr|
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