ARC239 dihydrochloride - CAS 67339-62-2
Catalog number:
67339-62-2
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C24H31Cl2N3O3
Molecular Weight:
480.43
COA:
Inquire
Targets:
Adrenergic Receptor
Description:
ARC239 dihydrochloride is a potent and selective α2 B adrenoceptor antagonist. It is used as an α-adrenoceptor blocking drug. It competitively antagonizes pressor responses to adrenaline and inhibits pressor responses to noradrenaline, tyramine, phenylephrine and dimethylphenylpiperazinium.
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Purity:
98%
Appearance:
Solid powder
Synonyms:
2-(2-(4-(2-Methoxyphenyl)piperazin-1-yl)ethyl)-4,4-dimethyl-1,3-(2H,4H)-isoquinolindione dihydrochloride;AR-C239 Dihydrochloride
Solubility:
Soluble in DMSO, not in water
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
ARC239 dihydrochloride is used as an α-adrenoceptor blocking drug.
Quality Standard:
In-house standard
Quantity:
Milligrams-Grams
Boiling Point:
595.8±50.0 °C | Condition: Press: 760 Torr
Density:
1.167±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
SAJKHRHHDGSJEZ-UHFFFAOYSA-N
InChI:
InChI=1S/C24H29N3O3.2ClH/c1-24(2)19-9-5-4-8-18(19)22(28)27(23(24)29)17-14-25-12-15-26(16-13-25)20-10-6-7-11-21(20)30-3;;/h4-11H,12-17H2,1-3H3;2*1H
Canonical SMILES:
CC1(C2=CC=CC=C2C(=O)N(C1=O)CCN3CCN(CC3)C4=CC=CC=C4OC)C.Cl.Cl
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CAS 67339-62-2 ARC239 dihydrochloride

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