AR-C 118925XX - CAS 216657-60-2
Category: Inhibitor
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Molecular Formula:
C28H23N7O3S
Molecular Weight:
537.59
COA:
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Targets:
P2Y Receptor
Description:
AR-C126313, a thiouracil derivative, has been found to be a competitive P2Y2 receptor antagonist and could inhibit P2Y2 receptor-induced β-arrestin translocation in vitro.
Purity:
≥97% by HPLC
Appearance:
Yellow Solid
Synonyms:
AR-C126313; ARC126313; AR C126313; 5-[[5-(2,8-Dimethyl-5H-dibenzo[a,d]cyclohepten-5-yl)-3,4-dihydro-2-oxo-4-thioxo-1(2H)-pyrimidinyl]methyl]-N-2H-tetrazol-5-yl-2-furancarboxamide
MSDS:
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InChIKey:
PVKNPGQAFNALOI-UHFFFAOYSA-N
InChI:
InChI=1S/C28H23N7O3S/c1-15-3-8-20-17(11-15)5-6-18-12-16(2)4-9-21(18)24(20)22-14-35(28(37)30-26(22)39)13-19-7-10-23(38-19)25(36)29-27-31-33-34-32-27/h3-12,14,24H,13H2,1-2H3,(H,30,37,39)(H2,29,31,32,33,34,36)
Canonical SMILES:
CC1=CC2=C(C=C1)C(C3=C(C=C2)C=C(C=C3)C)C4=CN(C(=O)NC4=S)CC5=CC=C(O5)C(=O)NC6=NNN=N6
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Chemical Structure

CAS 216657-60-2 AR-C 118925XX

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