AR-​08 - CAS 226081-74-9
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C12H12N6
Molecular Weight:
240.26
COA:
Inquire
Targets:
Adrenergic Receptor
Description:
AR-​08 is an agonist of α2-adrenergic receptor undergone in phase II clinical trials by Arbor Pharmaceuticals for the treatment of attention deficit and hyperactivity disorder (ADHD).
Publictions citing BOC Sciences Products
  • >> More
Synonyms:
6-(4,5-dihydro-1H-imidazol-2-ylamino)-7-methyl-3H-benzimidazole-4-carbonitrile; 1H-Benzimidazole-7-carbonitrile, 5-[(4,5-dihydro-1H-imidazol-2-yl)amino]-4-methyl-; 6-[(4,5-Dihydro-1H-imidazol-2-yl)amino-]-7-methyl-1H-benzimidazole-4-carbonitrile
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
545.2±60.0 ℃ at 760 Torr
Density:
1.50±0.1 g/cm3
InChIKey:
GONXJTJRZCPBLD-UHFFFAOYSA-N
InChI:
1S/C12H12N6/c1-7-9(18-12-14-2-3-15-12)4-8(5-13)11-10(7)16-6-17-11/h4,6H,2-3H2,1H3,(H,16,17)(H2,14,15,18)
Canonical SMILES:
CC1=C(C=C(C2=C1N=CN2)C#N)NC3=NCCN3
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related Adrenergic Receptor Products


CAS 5874-97-5 Metaproterenol hemisulfate salt

Metaproterenol hemisulfate salt
(CAS: 5874-97-5)

Metaproterenol hemisulfate salt is the hemisulfate salt form of Metaproterenol, which is a moderately selective beta-adrenergic agonist. It is used in the treat...

CAS 146-48-5 Yohimbine

Yohimbine
(CAS: 146-48-5)

Yohimbine, an indolalkylamine alkaloid, blocks presynaptic alpha-2 adrenergic receptors. IC50= 0.6 μM Ki: 1.05 nM, alphaα2Areceptor

CAS 849-55-8 Nylidrin hydrochloride

Nylidrin hydrochloride
(CAS: 849-55-8)

Nylidrin hydrochloride is a beta-adrenergic agonist. It was an effective inhibitor of IgE-mediated release of histamine from passively sensitized rat peritoneal...

CAS 661464-94-4 Levalbuterol tartrate

Levalbuterol tartrate
(CAS: 661464-94-4)

Levosalbutamol tartrate, the R-enantiomer of salbutamol, is a short-acting β2 adrenergic receptor agonist used in the treatment of asthma and chronic obstructiv...

CAS 38339-11-6 Clenproperol

Clenproperol
(CAS: 38339-11-6)

Clenproperol is a β-adrenergic agonist.

CAS 55974-42-0 ARC 239 dihydrochloride

ARC 239 dihydrochloride
(CAS: 55974-42-0)

The hydrochloride salt form of ARC 239, which has been found to be an α2B adrenoceptor antagonist as well as a norepinephrine-serotonin reuptake inhibitor.

CAS 1218-35-5 Xylometazoline HCl

Xylometazoline HCl
(CAS: 1218-35-5)

Xylometazoline is an α-adrenoceptor agonist commonly used as nasal decongestant, exhibits highest potency at α2B-adrenoceptor subtype with EC50 of 99 μM.

CAS 51384-51-1 Metoprolol

Metoprolol
(CAS: 51384-51-1)

Metoprolol is a a selective β1 receptor blocker for the treatment of a variety of cardiovascular disorder.

CAS 113145-69-0 (S)-(+)-Niguldipine hydrochloride

(S)-(+)-Niguldipine hydrochloride
(CAS: 113145-69-0)

(S)-(+)-Niguldipine hydrochloride, the more active enantiomer of Niguldipine hydrochloride, acts as a potent, selective α1A-adrenoceptor antagonist (Ki = 0.16 n...

CAS 157066-77-8 SNAP 5089

SNAP 5089
(CAS: 157066-77-8)

SNAP 5089 is an α1A-adrenoceptor antagonist with > 600-fold selectivity over other adrenoceptors (Ki = 0.35, 220, 370, 540, 800 and 1200 nM for α1A, α1B, α2C, α...

CAS 23076-35-9 Xylazine hydrochloride

Xylazine hydrochloride
(CAS: 23076-35-9)

Xylazine is an α2-Adrenergic receptor agonist, used as a sedative and muscle relaxant.It is used for sedation, anesthesia, muscle relaxation, and analgesia in a...

CAS 151126-84-0 CL 316243 disodium salt

CL 316243 disodium salt
(CAS: 151126-84-0)

The sodium salt form of CL 316243, which has been found to be a β3-adrenoceptor agonist and could probably decrease blood insulin as well as glucose levels.

CAS 964-52-3 Moxisylyte hydrochloride

Moxisylyte hydrochloride
(CAS: 964-52-3)

Moxisylyte hydrochloride is alpha 1-adrenoceptor antagonist. It can vasodilates cerebral vessels without reducing blood pressure. It is used as peripheral vasod...

CAS 36085-73-1 B-HT 920 dihydrochloride

B-HT 920 dihydrochloride
(CAS: 36085-73-1)

Talipexole is a D2 dopamine receptor agonist, displaying anti-Parkinsonian activity.

CAS 51022-70-9 Salbutamol Sulfate

Salbutamol Sulfate
(CAS: 51022-70-9)

Salbutamol Sulfate is a Non-selective 2-adrenergic receptor agonist (IC50=8.93 µM)

Fenoterol hydrochloride
(CAS: 1944-10-1)

Fenoterol hydrochloride is a β2 adrenoreceptor agonist used as a bronchodilator for the treatment and prophylaxis of reversible bronchospasm, administered by in...

Abanoquil mesilate
(CAS: 118931-00-3)

This molecular is an active biochemical as a Alpha 1 adrenergic receptor antagonist. However, no developments were reported for Ischaemic heart disorders and A...

CAS 13707-88-5 Alprenolol hydrochloride

Alprenolol hydrochloride
(CAS: 13707-88-5)

Alprenolol hydrochloride is the hydrochloride salt of alprenolol, which is a non-selective 5-HT1A receptor antagonist and beta blocker. It is used in the treatm...

CAS 200050-59-5 L-771688

L-771688
(CAS: 200050-59-5)

L-771688, also known as SNAP 6383, is a new potent and highly selective α1A-adrenoceptor antagonist with 500-fold selective over α1B and α1D-adrenoceptors.

CAS 94-07-5 Synephrine

Synephrine
(CAS: 94-07-5)

Synephrine is an α-adrenergic receptor agonist used as a vasoconstrictor.

Chemical Structure

CAS 226081-74-9 AR-​08

Quick Inquiry

Verification code

Featured Items