AP1903 - CAS 195514-63-7
Catalog number:
195514-63-7
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
COA:
Inquire
Targets:
Others
Description:
AP1903 is a lipid-permeable tacrolimus analogue with homodimerizing activity. Dimerizer drug AP1903 homodimerizes an analogue of human protein FKBP12 (Fv) which contains a single acid substitution (Phe36Val) so that AP1903 binds to wild-type FKBP12 with 1000-fold lower affinity.
Publictions citing BOC Sciences Products
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Purity:
0.98
Appearance:
Semisolid (wax like)
Synonyms:
AP 1903; AP-1903
MSDS:
Inquire
Current Developer:
ARIAD Pharm. / Bellicum Pharmaceuticals, Inc
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 195514-63-7 AP1903

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