|Description||Anpirtoline hydrochloride is the hydrochloride salt of anpirtoline, which is a highly potent 5-HT1B receptor agonist with Ki values of 28 nM. It decreases central serotonin synthesis and attenuates aggressive behavior in vivo. It also acts as an antagonist at 5-HT3 receptors with Ki value of 29.5 nM and is brain penetrant. It is a receptor agonist with antinociceptive/antidepressant-like actions in rodents.|
|Purity||≥99% by HPLC|
|Synonyms||6-Chloro-2-[piperidinyl-4-thio]pyridine hydrochloride; D16949; D-16949|
Tandospirone hydrochloride is a 5-HT1A receptor partial agonist (Ki = 27 nM) with selectivity over 5-HT2, 5-HT1C, α1, α2, D1 and D2 receptors (Ki values ranging...
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SB 216641 hydrochloride
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