Anpirtoline hydrochloride - CAS 99201-87-3
Category: Inhibitor
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Molecular Formula:
C10H14Cl2N2S
Molecular Weight:
265.20
COA:
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Targets:
5-HT Receptor
Description:
Anpirtoline hydrochloride is the hydrochloride salt of anpirtoline, which is a highly potent 5-HT1B receptor agonist with Ki values of 28 nM. It decreases central serotonin synthesis and attenuates aggressive behavior in vivo. It also acts as an antagonist at 5-HT3 receptors with Ki value of 29.5 nM and is brain penetrant. It is a receptor agonist with antinociceptive/antidepressant-like actions in rodents.
Purity:
≥99% by HPLC
Synonyms:
6-Chloro-2-[piperidinyl-4-thio]pyridine hydrochloride; D16949; D-16949
MSDS:
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InChIKey:
GRXDJABVNGUGCW-UHFFFAOYSA-N
InChI:
InChI=1S/C10H13ClN2S.ClH/c11-9-2-1-3-10(13-9)14-8-4-6-12-7-5-8;/h1-3,8,12H,4-7H2;1H
Canonical SMILES:
C1CNCCC1SC2=NC(=CC=C2)Cl.Cl
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Chemical Structure

CAS 99201-87-3 Anpirtoline hydrochloride

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