Anpirtoline hydrochloride - CAS 99201-87-3
Category: Inhibitor
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Molecular Formula:
Molecular Weight:
5-HT Receptor
Anpirtoline hydrochloride is the hydrochloride salt of anpirtoline, which is a highly potent 5-HT1B receptor agonist with Ki values of 28 nM. It decreases central serotonin synthesis and attenuates aggressive behavior in vivo. It also acts as an antagonist at 5-HT3 receptors with Ki value of 29.5 nM and is brain penetrant. It is a receptor agonist with antinociceptive/antidepressant-like actions in rodents.
≥99% by HPLC
6-Chloro-2-[piperidinyl-4-thio]pyridine hydrochloride; D16949; D-16949
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Chemical Structure

CAS 99201-87-3 Anpirtoline hydrochloride

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