|Description||(+)-Anabasine hydrochloride is a nicotine alkaloid present in tobacco products. It is a high affinity neuronal nicotinic ACh receptor partial agonist with Ki values of 0.058, 0.26 and 7.2 μM for rat α7, rat α4β2 and fish skeletal muscle nAChRs respectively. It also stimulates Ca2+-dependent catecholamine release from rat adrenomedullary cells in vitro. It is used as an indicator of smoking or tobacco use.|
|Purity||≥99% by HPLC|
Vecuronium bromide (Norcuron) is a muscle relaxant in the category of non-depolarizing blocking agents. Vecuronium bromide is indicated as an adjunct to general...
Cisatracurium besylate is a neuromuscular blocking agent that is used in liver transplant patient with safety. Cisatracurium besylate is also an enantiomer of A...
α-Conotoxin EI is a selective antagonist of neuromuscular nicotinic receptors α1β1γδ. It shows selectivity for α/δ sites over α/γ sites in Torpedo.
3-Bromocytisine has been found to be an α4β4, α4β2 and α7 nACh receptor agonist.
1-Acetyl-4-methylpiperazine hydrochloride is the hydrochloride salt of 1-Acetyl-4-methylpiperazine which is a structural analog of acetylcholine. It acts as a n...
TC 1698 dihydrochloride
TC 1698 dihydrochloride is a selective nicotinic α7 receptor agonist (EC50 = 440 nM) displaying neuroprotective activity. TC 1698 dihydrochloride also displays ...
A 582941 is a selective α7 nAChR partial agonist which is effetive for both rat and human α7 receptors (Ki = 10.8 and 16.7 nM respectively).
PHA 568487 is an orally active and brain penetrant agonist of the alpha 7 nicotinic acetylcholine receptor (Ki = 44 and 2800 for α7 and 5-HT3 respectively, IC50...