Amisulpride hydrochloride - CAS 81342-13-4
Catalog number: 81342-13-4
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C17H28N3O4SCl
Molecular Weight:
405.94
COA:
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Targets:
Dopamine Receptor
Description:
Amisulpride hydrochloride could inhibit radioligand binding to native dopamine D2 receptor in membranes from the rat striatum with an IC50 value of 21nM. It has been revealed to displace [3H]raclopride binding in vivo with an ED50 value of 17.3±1.86mg/kg in the rat limbic system. It has been noted to inhibit quinpirole-induced [3H]thymidine with an IC50 value of 22±3nM. It is used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder. It has been approved in February 2002 by FDA.
Purity:
>98%
Appearance:
Beige Solid
Synonyms:
DAN 2163 hydrochloride;4-amino-N-[(1-ethylpyrrolidin-2-yl)methyl]-5-ethylsulfonyl-2-methoxybenzamide;hydrochloride
Solubility:
DMSO 74 mg/mL ; Water <1 mg/mL ; Ethanol 74 mg/mL
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Amisulpride hydrochloride is used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder.
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
XFOYXFDTUMXXFP-UHFFFAOYSA-N
InChI:
InChI=1S/C17H27N3O4S.ClH/c1-4-20-8-6-7-12(20)11-19-17(21)13-9-16(25(22,23)5-2)14(18)10-15(13)24-3;/h9-10,12H,4-8,11,18H2,1-3H3,(H,19,21);1H
Canonical SMILES:
CCN1CCCC1CNC(=O)C2=CC(=C(C=C2OC)N)S(=O)(=O)CC.Cl
Current Developer:
Amisulpride hydrochloride It has been approved in February 2002 by FDA.
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