AMG8562 - CAS 1041478-78-7
Catalog number: 1041478-78-7
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C24H25F3N2O2
Molecular Weight:
430.47
COA:
Inquire
Targets:
TRP Channel
Description:
AMG8562 is a novel vanilloid receptor TRPV1 modulator.
Purity:
>98 %
Appearance:
Solid powder
Synonyms:
(E)-N-[(2R)-2-hydroxy-2,3-dihydro-1H-inden-4-yl]-3-[2-piperidin-1-yl-4-(trifluoromethyl)phenyl]prop-2-enamide;AMG-8562;2-Propenamide, N-((2R)-2,3-dihydro-2-hydroxy-1H-inden-4-yl)-3-(2-(1-piperidinyl)-4-(trifluoromethyl)phenyl)-, (2E)-
Solubility:
10 mM in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
Boiling Point:
617.8±55.0 °C | Condition: Press: 760 Torr
Density:
1.331±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
HAZYXDWNLMGLIS-LHUXKHBRSA-N
InChI:
InChI=1S/C24H25F3N2O2/c25-24(26,27)18-9-7-16(22(14-18)29-11-2-1-3-12-29)8-10-23(31)28-21-6-4-5-17-13-19(30)15-20(17)21/h4-10,14,19,30H,1-3,11-13,15H2,(H,28,31)/b10-8+/t19-/m1/s1
Canonical SMILES:
C1CCN(CC1)C2=C(C=CC(=C2)C(F)(F)F)C=CC(=O)NC3=CC=CC4=C3CC(C4)O
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