AMG319 - CAS 1608125-21-8
Catalog number: 1608125-21-8
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C21H16FN7
Molecular Weight:
385.4
COA:
Inquire
Targets:
PI3K
Description:
AMG319 is a potent and selective PI3Kδ inhibitor with IC50 of 18 nM, >47-fold selectivity over other PI3Ks. Phase 2.
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Purity:
98%
Appearance:
Solid powder
Synonyms:
AMG-319; AMG 319
Solubility:
DMSO,77mg/mL(199.79mM);Ethanol,77mg/mL(199.79mM);Water,<1mg/mL(<1mM)
Storage:
3 years -20℃powder;6 months-80℃in solvent
MSDS:
Inquire
Shelf Life:
2 years if stored properly
Canonical SMILES:
C[C@H](NC1=C2N=CNC2=NC=N1)C3=CC4=CC=C(F)C=C4N=C3C5=NC=CC=C5
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