AM095 (Free Acid) - CAS 1228690-36-5
Catalog number:
1228690-36-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C27H24N2O5
Molecular Weight:
456.49
COA:
Inquire
Targets:
LPL Receptor
Description:
AM095, an effective LPA1 receptor antagonist, has been found to decrease dermal fibrosis caused by attenuates bleomycin. IC50: 0.98 uM and 0.73 uM for human and mouse LPA1 respectively.
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Purity:
98%
Appearance:
Powder
Synonyms:
AM095 (free acid); CHEMBL2182052; AM095; AM-095 (free base); AM 095 (parent compound)
Solubility:
DMSO: ≥ 67.3 mg/mL
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
AM095 is an effective LPA1 receptor antagonist that has been found to decrease dermal fibrosis caused by attenuates bleomycin.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
LNDDRUPAICPXIN-GOSISDBHSA-N
InChI:
InChI=1S/C27H24N2O5/c1-17-25(28-27(32)33-18(2)20-6-4-3-5-7-20)26(34-29-17)23-14-12-22(13-15-23)21-10-8-19(9-11-21)16-24(30)31/h3-15,18H,16H2,1-2H3,(H,28,32)(H,30,31)/t18-/m1/s1
Canonical SMILES:
CC1=NOC(=C1NC(=O)OC(C)C2=CC=CC=C2)C3=CC=C(C=C3)C4=CC=C(C=C4)CC(=O)O
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