AM-9635 - CAS 1338483-10-5
Catalog number: 1338483-10-5
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C19H14F2N8
Molecular Weight:
392.36
COA:
Inquire
Targets:
PI3K
Description:
AM-9635 is a selective Phosphatidylinositol-3-kinase delta (PI3Kδ) inhibitor. AM-9635 exhibits good cellular potency (in vitro pAKT IC50 = 4.2 nM ). AM-9635 can inhibit KLH-specific IgG and IgM in a dosedependent manner and it is well tolerated at all doses. AM-96352 shows significantly reduced IgG and IgM specific antibodies.
Purity:
98%
Appearance:
Powder
Synonyms:
(S)-4-amino-6-((1-(6-fluoro-1-(5-fluoropyridin-3-yl)-1H-benzo[d]imidazol-2-yl)ethyl)amino)pyrimidine-5-carbonitrile
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
Boiling Point:
707.4±70.0 °C | Condition: Press: 760 Torr
Density:
1.52±0.1 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
Canonical SMILES:
N#CC1=C(N[C@H](C2=NC3=CC=C(F)C=C3N2C4=CC(F)=CN=C4)C)N=CN=C1N
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