Alosetron (Z)-2-butenedioate - CAS 122852-43-1
Catalog number:
122852-43-1
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C21H22N4O5
Molecular Weight:
410.42
COA:
Inquire
Targets:
5-HT Receptor
Description:
The maleic acid salt form of Alosetron which is an effective 5-HT3 receptor antagonist and could be commonly used against irritable bowel syndrome.
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Purity:
95%
Appearance:
Powder
Synonyms:
(Z)-but-2-enedioicacid;5-methyl-2-[(5-methyl-1H-imidazol-4-yl)methyl]-3,4-dihydropyrido[4,3-b]indol-1-one;Alosetron((Z)-2-butenedioate);122852-43-1;SCHEMBL1045;Alosetron(Z)-2-butenedioate
Solubility:
10 mM in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
The maleic acid salt form of Alosetron which is an effective 5-HT3 receptor antagonist and could be commonly used against irritable bowel syndrome.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
XCPGTDZMQXRLAW-BTJKTKAUSA-N
InChI:
InChI=1S/C17H18N4O.C4H4O4/c1-11-13(19-10-18-11)9-21-8-7-15-16(17(21)22)12-5-3-4-6-14(12)20(15)2;5-3(6)1-2-4(7)8/h3-6,10H,7-9H2,1-2H3,(H,18,19);1-2H,(H,5,6)(H,7,8)/b;2-1-
Canonical SMILES:
CC1=C(N=CN1)CN2CCC3=C(C2=O)C4=CC=CC=C4N3C.C(=CC(=O)O)C(=O)O
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Chemical Structure

CAS 122852-43-1 Alosetron (Z)-2-butenedioate

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