Aloisine B - CAS 496864-14-3
Catalog number: 496864-14-3
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C15H14ClN3
Molecular Weight:
271.75
COA:
Inquire
Targets:
CDK
Description:
Aloisine B is a potent and selective CDK and GSK-3 inhibitor with highest affinity targets: Glycogen Synthase Kinase-3, Beta (Rattus norvegicus (rat)) (IC50=750.0 nM).
Purity:
≥98%
Appearance:
Yellow solid
Synonyms:
6-(4-chlorophenyl)-7-(propan-2-yl)-5H-pyrrolo[2,3-b]pyrazine; 6-phenyl[5H]pyrrolo[2,3-b]pyrazine (aloisine) 37; 6-(4-chlorophenyl)-7-isopropyl-5H-pyrrolo[2,3-b]pyrazine;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
A potent and selective CDK and GSK-3 inhibitor.
Quality Standard:
Enterprise Standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly.
Quantity:
Milligrams-Grams
InChIKey:
GFJIABMYYUGNEC-UHFFFAOYSA-N
InChI:
1S/C15H14ClN3/c1-9(2)12-13(10-3-5-11(16)6-4-10)19-15-14(12)17-7-8-18-15/h3-9H,1-2H3,(H,18,19)
Canonical SMILES:
CC(C1=C(C2=CC=C(Cl)C=C2)NC3=NC=CN=C31)C
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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