|Description||Allopurinol Sodium is a xanthine oxidase inhibitor with an IC50 of 7.82±0.12 μM.|
MLN1117, also known as INK1117, is a PI3Kα inhibitor which could lead to the apoptosis and growth retardation of tumor cells expressed by PI3Kα. IC50: 15 nM.
L-655,708, an inverse agonist of α5 subunit involved in GABAA receptor, has been found to exhibit cognitive performance improvement in biological studies.
Thioperamide is a potent histamine H3 and H4 antagonist/inverse agonist (Ki = 25 and 27 nM for human recombinant H3 and H4 receptors, respectively). Thioperamid...
L-trans-2,4-PDC is a competitive, transportable inhibitor of L-glutamate transport (Ki = 4.6 μM in rat brain synaptosomes).
DPC AJ1951 has been found to be a potent agonist of the PTH/PTH-related peptide receptor.
Ozanimod, also known as RPC1063, is a selective oral S1P Receptor 1 modulator.
IKK-2 inhibitor VIII
IKK-2 inhibitor VIII is a potent and selective IKK-2 inhibitor.
MK-0893 is a selective glucagon receptor antagonist. It can block glucagon binding to the human GCGR and antagonize glucagon-induced intracellular accumulation ...