|Description||Alfuzosin HCl is an alpha1 receptor antagonist used to treat benign prostatic hyperplasia (BPH).|
This molecular is an active biochemical as a Alpha 1 adrenergic receptor antagonist. However, no developments were reported for Ischaemic heart disorders and A...
Indacaterol is an ultra-long-acting β-adrenoceptor agonist with pKi of 7.36.
MK-761 has beta adrenoceptor antagonist and vasodilating properties in a single molecule. It has beta adrenoceptor blocking activity in the isolated cat heart p...
Sotalol hydrochloride is a non-selective beta adrenoceptor antagonist and potassium channel blocker (IC50 = 43 μM)
Tertatolol, a benzothiopyran derivative, is a potent dual antagonist of beta-adrenoceptor and 5-HT receptor, with antihypertensive effect.
Aptazapine is a tetracyclic antidepressant. It was assayed in clinical trials for the treatment of depression in the 1980s but was never marketed. Aptazapine is...
Tetrahydrozoline HCl is an imidazoline derivative with alpha receptor agonist activity.
Setiptiline is is a serotonin receptor antagonist acts as a noradrenergic and specific serotonergic antidepressant.
Tamsulosin could block on the sympathetic α1 receptor, especially selectively bind to the α1A receptor and has been found to be effective in the treatment of be...
D2343 is a dual inhibitor of β2-adrenoceptor and α1- adrenoceptor. Inhaled D2343 has a longer bronchodilating effect than terbutaline.
Betaxolol is a β1 adrenergic receptor blocker with IC50 of 6 μM.
Fenmetozole, also known as DH-524, is an antagonist of α2-adrenergic receptor and also antagonizes the actions of ethanol.
BMS-194449 was found to be a β-adrenergic receptor agonist that was once studied in antihyperglycaemics as well as obesity therapy.
Deoxycorticosterone acetate is a steroid hormone used for intramuscular injection for replacement therapy of the adrenocortical steroid.
Salbutamol Sulfate is a Non-selective 2-adrenergic receptor agonist (IC50=8.93 µM)
Milveterol is a long-acting β(2)-adrenoceptor agonist under the development of GlaxoSmithKline. Phase II trials for the treatment of Chronic obstructive pulmona...
Brimonidine is α2-Adrenoceptor agonist. It is a drug used as eye drops to treat open-angle glaucoma or ocular hypertension. It acts via decreasing synthesis of ...
BMS-196085, a sulfanilamide derivative, has been found to be a β-adrenergic receptor agonist that was once studied in obesity as well as yype 2 diabetes mellitu...
Pirbuterol acetate is a short-acting β2 adrenoreceptor agonist. It has bronchodilating action and is used as a bronchodilator. It is also used in the treatment ...
Levosalbutamol tartrate, the R-enantiomer of salbutamol, is a short-acting β2 adrenergic receptor agonist used in the treatment of asthma and chronic obstructiv...