Agomelatine hydrochloride - CAS 1176316-99-6
Catalog number:
1176316-99-6
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C15H18ClNO2
Molecular Weight:
279.76
COA:
Inquire
Targets:
5-HT Receptor
Description:
The hydrochloride salt form of Agomelatine that is an antidepressant agent for acting as an antagonism of the 5-HT2C receptor. It is also an antagonist of 5-HT2B receptors. IC50: 6.2 and 6.6 for 5-HT2c and 5-HT2b respectively (pKi ).
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Purity:
98%
Appearance:
Powder
Synonyms:
Valdoxan hydrochloride; S-20098 hydrochloride
Solubility:
DMSO 49 mg/mL ; Water <1 mg/mL ; Ethanol 49 mg/mL
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
The hydrochloride salt form of Agomelatine that is an antidepressant agent for acting as an antagonism of the 5-HT2C receptor.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
ZJVMEXOLMFNQPX-UHFFFAOYSA-N
InChI:
InChI=1S/C15H17NO2.ClH/c1-11(17)16-9-8-13-5-3-4-12-6-7-14(18-2)10-15(12)13;/h3-7,10H,8-9H2,1-2H3,(H,16,17);1H
Canonical SMILES:
CC(=O)NCCC1=CC=CC2=C1C=C(C=C2)OC.Cl
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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