|Description||AF38469 is a novel, selective, orally bioavailable Sortilin inhibitor and showed no inhibition or stimulation of >50% at 10μM in a standard selectivity panel of ca. 70 targets run at CEREP. AF38469 showed no activity against the NTR1 receptor. In addition|
|Synonyms||2-[(6-methylpyridin-2-yl)carbamoyl]-5-(trifluoromethyl)benzoic acid CHEMBL3098745 AF38469 4n7e SCHEMBL15903106 BDBM50445054 ZINC95921158 HY-12802 KB-274741 n-(6-methylpyridin-2-yl)-5-trifluoromethyl-phthalamic acid|
|Solubility||Soluble to ≥ 43 mg/mL in DMSO|
|Storage||Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -63℃ for long term (months to years).|
|Shelf Life||2 years|
|Boiling Point||392.3±42.0 °C | Condition: Press: 760 Torr|
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