|Description||Aderbasib is a sheddase inhibitor, is also an orally bioavailable inhibitor of the ADAM (A Disintegrin And Metalloprotease) family of multifunctional membrane-bound proteins with potential antineoplastic activity. Aderbasib represses the metalloproteinase "sheddase" activities of ADAM10 and ADAM17, which may result in the inhibition of tumor cell proliferation.|
Diclofenac diethylamine is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.
GSK 789472 hydrochloride
GSK 789472 hydrochloride is a selective dopamine D3 receptor antagonist and D2 partial agonist (pEC50 values are <5.5 and 8.3, respectively). GSK 789472 exhibit...
R1487 is an orally bioavailable and highly selective inhibitors of p38α mitogen-activated protein kinase. (last upddated: 3/24/2016)
Arecaidine But-2-ynyl Ester Tosylate (ABET) is a potent and selective agonist of M2 recceptors in the atrium versus those in the ileum.
IPAG is a potent NMDA receptor antagonist at σ sites. It was used as an old antipsychiatric.
MNI-caged-D-aspartate, a photolabelled derivative of D-aspartate, is photolyzed by UV light with a quantum efficiency of 0.09 at pH 7.4. MNI-caged-D-aspartate i...
Psoralen is an active ingredient from Fructus Psoraleae and has anticancer activity.
MS 245 oxalate
MS 245 oxalate is a 5-HT6 antagonist with high affinity (Ki = 2.1 nM). It potentiates the hypolocomotor actions of (-)-nicotine in mice.