ACT 335827 - CAS 1354039-86-3
Category: Inhibitor
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Molecular Formula:
C31H38N2O5
Molecular Weight:
518.64
COA:
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Targets:
Orexin Receptor (OX Receptor)
Description:
ACT 335827 has been found to be an orexin OX1 receptor antagonist and could probably exhibit anxiolytic effects in vivo.
Purity:
≥98% by HPLC
Appearance:
Off-white Solid
Synonyms:
ACT-335827; ACT 335827; ACT335827; (aR,1S)-1-[(3,4-Dimethoxyphenyl)methyl]-3,4-dihydro-6,7-dimethoxy-N-(1-methylethyl)-a-phenyl-2(1H)-isoquinolineacetamide
MSDS:
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InChIKey:
HXHOBPVRRPCTLG-SETSBSEESA-N
InChI:
InChI=1S/C31H38N2O5/c1-20(2)32-31(34)30(22-10-8-7-9-11-22)33-15-14-23-18-28(37-5)29(38-6)19-24(23)25(33)16-21-12-13-26(35-3)27(17-21)36-4/h7-13,17-20,25,30H,14-16H2,1-6H3,(H,32,34)/t25-,30+/m0/s1
Canonical SMILES:
CC(C)NC(=O)C(C1=CC=CC=C1)N2CCC3=CC(=C(C=C3C2CC4=CC(=C(C=C4)OC)OC)OC)OC
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Chemical Structure

CAS 1354039-86-3 ACT 335827

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