|Description||This molecular is a prodrug of ACT-246475 which is a selective P2Y12 receptor antagonist with a wider therapeutic window in the rat model. ACT-281959 is the phosphate of ACT-246475 and showed antithrombotic efficacy after oral administration in the rat ferric chloride model. In May 2016, Phase-I development is ongoing in France.|
|Solubility||Soluble in DMSO|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
|Current Developer||Originator:Actelion Pharmaceuticals|
This active molecular is an immunoactive substance that produced by Paecilomyces carneus F-4882, an imperfect fungus. FR-901235 can lead to the mitogen-induced ...
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