|Description||This molecular is a prodrug of ACT-246475 which is a selective P2Y12 receptor antagonist with a wider therapeutic window in the rat model. ACT-281959 is the phosphate of ACT-246475 and showed antithrombotic efficacy after oral administration in the rat ferric chloride model. In May 2016, Phase-I development is ongoing in France.|
|Solubility||Soluble in DMSO|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
|Current Developer||Originator:Actelion Pharmaceuticals|
Cinobufotalin is one of the bufadienolides prepared from toad venom. It has anticancer activity.
Edaravone is a novel potent free radical scavenger that reduces reactive oxygen species, inhibites apoptosis, and blocks nonenzymatic peroxidation and lipoxygen...
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Extract from Aconitum carmichaeli Debx.
Propanil is a widely used contact herbicide mainly used to control weed growth in rice fields.
Nicotinic acid N-oxide
Nicotinic acid N-oxide is used to treat hyperlipoidemia.
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Tiaprofenic acid is a non-steroidal anti-inflammatory drug used to treat pain, especially arthritic pain.
A Metabolite of Pomalidomide.
Carbinoxamine is a antihistamine and anticholinergic agent used in the treatment of severe itching in patients with CD5.
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AKBA is an active triterpenoid compound from the extract of Boswellia serrate and a novel Nrf2 activator.
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