|Description||This active molecular is a reversible and selective platelet P2Y12 receptor antagonist. IC50 value of ACT-246475 is 8.0 nM. ACT-246475 dose-dependently blocked thrombus formation in the rat ferric chloride model and displayed a wide therapeutic window. In May 2016, Phase-I development is ongoing in France.|
|Solubility||Soluble in DMSO|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
|Current Developer||Originator:Actelion Pharmaceuticals|
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