ACT 178882 - CAS 1007392-69-9
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C33H38Cl3N3O4
Molecular Weight:
647.03
COA:
Inquire
Targets:
Renin
Description:
ACT 178882 is a novel Renin inhibitor (IC50= 1.4 nM).
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Synonyms:
(3R,4S)-N-[[2-chloro-5-(2-methoxyethyl)phenyl]methyl]-N-cyclopropyl-4-[6-[2-(2,6-dichloro-4-methylphenoxy)ethoxy]pyridin-3-yl]piperidine-3-carboxamide
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
764.3±60.0 ℃ at 760 Torr
Density:
1.33±0.1 g/cm3
InChIKey:
PGSRKJVMAOWDEC-SXOMAYOGSA-N
InChI:
1S/C33H38Cl3N3O4/c1-21-15-29(35)32(30(36)16-21)43-14-13-42-31-8-4-23(18-38-31)26-9-11-37-19-27(26)33(40)39(25-5-6-25)20-24-17-22(10-12-41-2)3-7-28(24)34/h3-4,7-8,15-18,25-27,37H,5-6,9-14,19-20H2,1-2H3/t26-,27+/m1/s1
Canonical SMILES:
CC1=CC(=C(C(=C1)Cl)OCCOC2=NC=C(C=C2)C3CCNCC3C(=O)N(CC4=C(C=CC(=C4)CCOC)Cl)C5CC5)Cl
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 1007392-69-9 ACT 178882

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