aceprometazine - CAS 13461-01-3
Catalog number: 13461-01-3
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H22N2OS
Molecular Weight:
326.46
COA:
Inquire
Targets:
Histamine Receptor
Description:
Aceprometazine is a Histamine H1 receptor antagonist as an approved drug. It can be used in combination with meprobamate for the treatment of sleep disorders such as Insomnia.
Publictions citing BOC Sciences Products
  • >> More
Purity:
95%
Appearance:
Powder
Synonyms:
aceprometazine;1-[10-[2-(Dimethylamino)propyl]-10H-phenothiazin-2-yl]ethanone;Acepromethazine
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Insomnia
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
Boiling Point:
490.1ºC at 760mmHg
Density:
1.154g/cm3
InChIKey:
XLOQNFNTQIRSOX-UHFFFAOYSA-N
InChI:
InChI=1S/C19H22N2OS/c1-13(20(3)4)12-21-16-7-5-6-8-18(16)23-19-10-9-15(14(2)22)11-17(19)21/h5-11,13H,12H2,1-4H3
Canonical SMILES:
CC(CN1C2=CC=CC=C2SC3=C1C=C(C=C3)C(=O)C)N(C)C
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related Histamine Receptor Products


CAS 76239-32-2 KP136

KP136
(CAS: 76239-32-2)

KP136, an antiallergic agent, remarkably inhibited the passive cutaneous anaphylaxis (PCA) with intravenous and oral dosing. KP-136 is an oral potent inhibitor ...

CAS 14976-57-9 Clemastine Fumarate

Clemastine Fumarate
(CAS: 14976-57-9)

Clemastine Fumarate (Clemastine) is a selective histamine H1 receptor antagonist with IC50 of 3 nM.

FR-A 19
(CAS: 141099-46-9)

FR-A 19 is a Histamine H2 receptor agonist with potent anti-allergic properties. It can inhibit IgE-mediated human basophil histamine release in a nanomolar ran...

CAS 1163-36-6 Clemizole hydrochloride

Clemizole hydrochloride
(CAS: 1163-36-6)

The hydrochloride salt form of Clemizole that has hepatitis C antiviral effect through restraining NS4B function and could also be used as an anticonvulsant in ...

CAS 6153-33-9 Mebhydroline Napadisylate

Mebhydroline Napadisylate
(CAS: 6153-33-9)

Mebhydroline Napadisylate is an antihistamine used for symptomatic relief of allergic symptoms caused by histamine release, including nasal allergies and allerg...

CAS 21535-47-7 Mianserin Hydrochloride

Mianserin Hydrochloride
(CAS: 21535-47-7)

Mianserin Hydrochloride is a psychoactive drug of the tetracyclic antidepressant.It is classified as a noradrenergic and specific serotonergic antidepressant (N...

LY-150310
(CAS: 103294-47-9)

LY-150310 is a histamine H1-receptor antagonist. It could alter prostanoid concentrations in vitro and in vivo.

GS-283
(CAS: 149440-36-8)

GS-283, an isoquinolin derivative, has been found to be histamine receptor and muscarinic receptor blocker.

CAS 3964-81-6 Azatadine

Azatadine
(CAS: 3964-81-6)

Azatadine is a new antihistamine acts as histamine for histamine H1- receptor inhibitor ( IC50 = 6.5 nM and 10 nM, respectively).

CAS 73903-17-0 JNJ-10191584

JNJ-10191584
(CAS: 73903-17-0)

JNJ-10191584 is a selective histamine H4 receptor antagonist. It inhibits mast cell in vitro with IC50 value of 138nM. JNJ-10191584 has antiinflammatory and ana...

CAS 83799-24-0 Fexofenadine

Fexofenadine
(CAS: 83799-24-0)

Fexofenadine is Histamine H1 receptor antagonist. It can be used for the treatment of allergy symptoms, such as hay fever, nasal congestion, and urticaria.

CAS 51-45-6 Histamine

Histamine
(CAS: 51-45-6)

Histamine is an organic nitrogenous compound produced by basophils and by mast cells found in nearby connective tissues.

CAS 2192-20-3 Hydroxyzine dihydrochloride

Hydroxyzine dihydrochloride
(CAS: 2192-20-3)

Hydroxyzine (sold as Vistaril, Atarax) is a first-generation antihistamine of the diphenylmethane and piperazine class.

CAS 132-20-7 Pheniramine Maleate

Pheniramine Maleate
(CAS: 132-20-7)

Pheniramine Maleate is an antihistamine with anticholinergic properties used to treat allergic conditions such as hay fever or urticaria.

CAS 84-96-8 Trimeprazine

Trimeprazine
(CAS: 84-96-8)

Alimemazine is a phenothiazine derivative as a Histamine Receptor antagonist. It can be used as an antipruritic . It also acts as a sedative, hypnotic, and anti...

CAS 113-69-9 Benzquinamide Hydrochloride

Benzquinamide Hydrochloride
(CAS: 113-69-9)

Benzquinamide hydrochloride is an antiemetic compound with antihistaminic, anticholinergic and sedative properties. The mechanism of action is not quite sure an...

CAS 77-38-3 Chlorphenoxamine

Chlorphenoxamine
(CAS: 77-38-3)

Chlorphenoxamine is an analog of diphenhydramine. It has antimuscarinic and antihistaminic properties. It has been used as an antipruritic and antiparkinsonian ...

SUVN-G3031 hydrochloride
(CAS: 1394808-20-8)

SUVN-G3031 is a Histamine H3 receptor antagonist originated by Suven Life Sciences. Blockade of Histamine H3 receptor can augment the pre-synaptic release of bo...

CAS 3978-86-7 Azatadine dimaleate

Azatadine dimaleate
(CAS: 3978-86-7)

Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.

CAS 76963-41-2 Nizatidine

Nizatidine
(CAS: 76963-41-2)

Nizatidine is a histamine H2 receptor antagonist with IC50 of 0.9 nM, also inhibits AChE with IC50 of 6.7 μM.

Chemical Structure

CAS 13461-01-3 aceprometazine

Quick Inquiry

Verification code

Featured Items