|Description||A selective FAP inhibitor (Ki= 23 nM)|
|Storage||Store in a cool and dry place (or refer to the Certificate of Analysis).|
Tofisopam, a 2,3-benzodiazepine, has depressant effects at high doses in several different animal test procedures. Tofisopam has been shown to enhance the antic...
Aminohippurate Sodium is a diagnostic agent that is used to help differentiate and characterized organic anion transporter (OAT) isoforms. It is useful in medic...
Acetyl-Calpastatin (184-210) (human)
Acetyl-Calpastatin (184-210) (human) is a calpain I/II inhibitor and could increase secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio.
Glutapyrone is a DHP amino acid used in the antiarrhythmic, neuroprotective, stress-protective and radioprotective remedy.
TCS 3035 is a GPR35 agonist (pEC50 = 5.13 and 5.86 for rat and human GPR35 orthologs, respectively).
BMS-243117 is a potent and selective Lck inhibitor with good cellular activity against T-cell proliferation. BMS-24311 has potential to treat diseases such as r...
Methylmalonate, a dicarboxylic acid that can be derived from methylmalonyl-coenzyme A (methylmalonyl-CoA), binds with coenzyme A to form methylmalonyl-CoA. It i...
TP 064 is a potent and selective PRMT4 inhibitor with >100-fold selectivity over other histone methyltransferases and non-epigenetic targets. TP 064 inhibits me...
Diacerin is an inhibitor of pro-inflammatory cytokine Interleukin-1B (IL-1B) production, prescribed for osteoarthritis and chronic inflammatory arthritis.
Carboxy-PTIO, potassium salt
The potassium salt form of Carboxy-PTIO, which is a water soluble, stable organic free radical that could react stoichiometrically with NO.
FR-193262 is a designed prostacyclin mimetic without PG skeleton which exhibits potent PGI2 agonistic activity with good selectivity for IP receptor and bioavai...
Pseudobufarenogin is a natural compound extracted from toad species with unknown details.
PPNDS is a potent and selective P2X1 receptor antagonist (pKB = 7.43 in rat vas deferens). PNDS is approximately 50-fold less selective for P2Y1R and does not i...
Auranofin appears to induce heme oxygenase 1 (HO-1) mRNA, as an inhibitor of thioredoxin reductase (TrxR) (IC50 = 20 nM; Ki = 4 nM for the NADPH-reduced form of...
β-Apo-13-carotenone, also known as D'Orenone, a naturally occurring β-apocarotenoid, is an antagonist of RXRα.
N-Acetylglycyl-D-glutamic acid is a kind of excitatory peptide. It is more potent than L-glutamic acid at inducing seizures in mice.
Arg-Gly-Asp-Cys is the binding motif of fibronectin to cell adhesion molecules, and surfaces modified with RGDC were shown to be effective for osteoblast bindin...
Imidazole, a highly polar compound, has been used extensively as a corrosion inhibitor and a buffer in the pH range of 6.2-7.8.
Etimizol was shown to relieve amnesia effectively in the origin of which there is the hypoxic component (hypobaric hypoxia, actinomycin D, mechanical injury of ...
CGP 20376 is a benzothiazole compound and it has antifilarial properties.