|Description||A selective FAP inhibitor (Ki= 23 nM)|
|Storage||Store in a cool and dry place (or refer to the Certificate of Analysis).|
Acetyl-Calpastatin (184-210) (human)
Acetyl-Calpastatin (184-210) (human) is a calpain I/II inhibitor and could increase secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio.
Ocaphane Hydrochloride is a strong antitumor agent used on a number of animal tumors such as Brown-Pearce carcinoma but is fairly toxic to hemopoietic organs.
Ouabain is a cardiac glycoside acting by Na(+)/K(+) ATPase, regulates transcription of MDR and MRP.
Carbimazole is used to treat hyperthyroidism. Carbimazole is a pro-drug as after absorption it is converted to the active form, methimazole. Methimazole prevent...
Aladorianis is a ryanodine receptor calcium release channel modulator. It is an antiarrhythmic agent. Clinical development for Chronic heart failure and Ventric...
CaCCinh-A01 has been found to be a calcium-activated chloride channel (CaCC) inhibitor, wich IC50 ~ 10 μM.
A 1120 is a retinol-binding protein 4 (RBP4) antagonist (Ki = 8.3 nM) that can reduce serum RBP4 and retinol, and displaces transthyretin (TTR) from RBP4-TTR co...
Fanetizole shows immunoregulating activity.