|Description||Abiraterone blocks the synthesis of androgens by inhibiting CYP17A1. It is used to treat metastatic, castration-resistant prostate cancer.|
|B0084-059670||5 g||$198||In stock|
|Brife Description||CYP17A1 inhibitor, metastatic, castration-resistant prostate cancer|
|Synonyms||(3beta)-17-(3-pyridinyl)-androsta-5,16-dien-3-ol; 17-(3-Pyridyl)androsta-5,16-dien-3beta-ol; CB 7598; CB-7598|
|Application||the treatment of metastatic, castration-resistant prostate cancer|
Abiraterone blocks the synthesis of androgens by inhibiting CYP17A1. It is used to treat metastatic, castration-resistant prostate cancer.
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The acetate form of abiraterone, which blocks the synthesis of androgens by inhibiting CYP17A1.
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VT-464 R enantiomer
The R-enantiomer form of VT-464, a non-steroidal compound, has been found to lead to the reduction of androgen through acting as a human CYP17 lyase inhibitor.
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The racemate form of VT-464, a non-steroidal compound, has been found to lead to the reduction of androgen through acting as a human CYP17 lyase inhibitor. IC50...