A-77-01 - CAS 607737-87-1
Catalog number:
607737-87-1
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C18H14N4
Molecular Weight:
286.34
COA:
Inquire
Targets:
TGF-β Receptor
Description:
A-77-01 is an inhibitor of TGF-β type I receptor superfamily activin-like kinase ALK5( IC50 =25nM).
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Purity:
≥98%
Appearance:
Light yellow to yellow solid
Synonyms:
4-[3-(6-Methyl-2-pyridinyl)-1H-pyrazol-4-yl]-quinoline; 4-[3-(6-Methyl-pyridin-2-yl)-1H-pyrazol-4-yl]-quinoline;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
Potent ALK5 inhibitor
Quality Standard:
Enterprise Standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
KJTYZDORHCDZPS-UHFFFAOYSA-N
InChI:
1S/C18H14N4/c1-12-5-4-8-17(21-12)18-15(11-20-22-18)13-9-10-19-16-7-3-2-6-14(13)16/h2-11H,1H3,(H,20,22)
Canonical SMILES:
CC1=CC=CC(=N1)C2=C(C=NN2)C3=CC=NC4=CC=CC=C34
Current Developer:
Sanofi-aventis
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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Chemical Structure

CAS 607737-87-1 A-77-01

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