A 582941 - CAS 848591-90-2
Category: Inhibitor
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Molecular Formula:
C17H20N4
Molecular Weight:
280.37
COA:
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Targets:
nAChR
Description:
A 582941 is a selective α7 nAChR partial agonist which is effetive for both rat and human α7 receptors (Ki = 10.8 and 16.7 nM respectively).
Brife Description:
α7 nAChR partial agonist
Purity:
≥98% by HPLC
Synonyms:
A-582941; Octahydro-2-methyl-5-(6-phenyl-3-pyridazinyl)-pyrrolo[3,4-c]pyrrole; (3aR,6aS)-2-methyl-5-(6-phenylpyridazin-3-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole
MSDS:
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InChIKey:
GTMRUYCIJSNXGB-GASCZTMLSA-N
InChI:
InChI=1S/C17H20N4/c1-20-9-14-11-21(12-15(14)10-20)17-8-7-16(18-19-17)13-5-3-2-4-6-13/h2-8,14-15H,9-12H2,1H3/t14-,15+
Canonical SMILES:
CN1CC2CN(CC2C1)C3=NN=C(C=C3)C4=CC=CC=C4
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Chemical Structure

CAS 848591-90-2 A 582941

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