|Description||A-366 is peptide-competitive inhibitor of the G9a/GLP histone lysine methyltransferase (IC50 = 3.3 nM) and is approximately 1,000-fold selective over other methyltransferases.|
|Synonyms||5'-methoxy-6'-(3-pyrrolidin-1-ylpropoxy)spiro[cyclobutane-1,3'-indole]-2'-amine A-366 CHEMBL3109630 A 366 GTPL8238 SCHEMBL17106564 BDBM50446376 ZINC95921314 AKOS024458525 CS-4644 HY-12583 B4947 5'-methoxy-6'-[3-(pyrrolidin-1-yl)propoxy]spiro[cyclobutane-1|
|Solubility||Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO|
|Storage||Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -57℃ for long term (months to years).|
|Shelf Life||2 years|
|Boiling Point||533.6±60.0 °C | Condition: Press: 760 Torr|
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