|Description||6'-Iodoresiniferatoxin is a partial and high affinity TRPV1 (VR1) vanilloid receptor agonist with EC50 value of 130 nM and Ki value of 0.71 nM. It shows partial agonism at human VR1 and full agonism at rat VR1.|
|Purity||≥98% by HPLC|
|Synonyms||6'-IRTX; [(2S,3aR,3bS,6aR,9aR,9bR,10R,11aR)-3a,3b,6,6a,9a,10,11,11a-octahydro-6a-hydroxy-8,10-dimethyl-11a-(1-methylethenyl)-7-oxo-2-(phenylmethyl)-7H-2,9b-epoxyazuleno[5,4-e]-1,3-benzodioxol-5-yl]-4-hydroxy-2-iodo-5-methoxy-benzeneacetic acid methyl ester|
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