6'-GNTI dihydrochloride
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C27H29N5O3.2HCl
Molecular Weight:
544.48
COA:
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Targets:
Opioid Receptor
Description:
6'-GNTI dihydrochloride is a potent and selective κ/δ-opioid heterodimer receptor agonist (EC50 = 39.8, 112.5 and > 1000 nM for κ/δ, κ/μ and δ/μ, respectively) without effecting on opioid receptor homodimers (EC50 > 1000 nM). 6'-GNTI exhibits tissue-specific analgesic effects in vitro.
Brife Description:
κ/δ-opioid heterodimer receptor agonist
Purity:
≥97% by HPLC
Synonyms:
6''-Guanidinyl-17-(cyclopropylmethyl)-6,7-dehydro-4,5a-epoxy-3,14-dihydroxy-6,7-2',3'-indolomorphinan dihydrochloride
MSDS:
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